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Somatostatin analog · octapeptide

Octreotide

/ok-TREE-oh-tide/FDA-approved ingredient
Interactive anatomyExplore where this peptide acts.

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At a glance

What is it—and why does it matter?

Octreotide is a cyclic peptide made of eight amino acids with long-acting somatostatin-like pharmacologic activity. Octreotide is reported as a full agonist at the human somatostatin SST5 receptor, with binding affinity expressed as pKi 7.2 - 9.5. In a two-case neonatal report of mutation-associated hypoglycemia (KCNJ11/ABCC8; congenital hyperinsulinism), octreotide administration was associated with stabilization of glycemic levels, after failure of enteral/parenteral glucose infusions and lack of clinical response to diazoxide. The labeled contraindication is allergy/hypersensitivity to the active peptide (octreotide) or excipients in MYCAPSSA, reflecting risk of serious allergic reactions.

Evidence behind this overview

Each sentence above is copied from a published claim presentation. The links open its evidence record.

ClassSomatostatin analog
Structure8 amino acids
StatusFDA-approved ingredient
Products in this profile3
The important boundary

Indication and transition instructions depend heavily on immediate-release, depot, or oral formulation. [1]Regulatory labelSandostatin prescribing informationCurrent DailyMed immediate-release octreotide label.

Identity + structure

A molecule, not a product name.

Chemical identity and product identity are kept separate so evidence does not leak between formulations or indications.
Preferred nameOctreotideIngredient
Pharmacologic classSomatostatin analogProfile record
Peptide structure8 amino acidsProfile record
Also indexed asoctreotide · octreotide acetate · somatostatin analogSearch aliases

Mechanism + clinical pharmacology

Target, response, and disposition.

Primary explanation

Suppresses growth hormone and multiple gastrointestinal/pancreatic hormones through somatostatin receptors. [1]Regulatory labelSandostatin prescribing informationCurrent DailyMed immediate-release octreotide label.

Evidence ledger

What the evidence says.

301 profile findings. Contextual and unclassified research is listed separately below. Open each citation to inspect the source and its limitations.

These are evidence statements, not individualized medical instructions. Product, dose, population, and study context remain attached to each source.

Study findings

What studies observed in defined populations, comparators, and time periods.

62 statements
Source-backed statement

CHEMBL1680 bound the human SST2 receptor with Ki = 0.4 nM.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

When PRRT eligibility was defined by NETTER-1 (Krenning ≥2), more patients met eligibility on PET than on planar imaging performed with [111In]octreotide scintigraphy.

Sources[63]Published evidence snapshotComparison of [111In]octreotide Scintigraphy and [68Ga]DOTATOC PET in Gastroenteropancreatic Neuroendocrine Tumors: Concordance of Krenning Scores and Implications for Peptide Receptor Radionuclide Therapy Eligibility.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The reported overall incidence of delayed bleeding in the cohort was 20% (21 events among 107).

Sources[56]Published evidence snapshotOctreotide for prevention of delayed bleeding after endoscopic mucosal resection for large superficial non-ampullary duodenal tumors.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The 18 F-octreotide PET/CT demonstrated concordant high tracer uptake in lesions that corresponded to lesions with intense uptake on 18 F-FDG PET/CT in this case.

Sources[61]Published evidence snapshotpubmed-42029102pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The review analyzed 33 children with an average age of 6.3 years.

Sources[72]Published evidence snapshotEfficacy and Safety of Octreotide for Gastrointestinal Bleeding Due to Portal Hypertension in Children-A Systematic Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a retrospective multi-center chart review, post-initiation hypoglycemia frequency differed by octreotide route: IV infusion had a higher median count than IV bolus or subcutaneous administration.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In the analyzed group (n=28), octreotide scintigraphy was positive in 71.4% and negative in 28.6%, and all positive scans were graded as mild uptake.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The evidence summarized does not support a consensus recommendation for when to initiate octreotide in adult chylothorax.

Sources[46]Published evidence snapshot[Optimal timing for octreotide administration in adult patients with chylothorax: A scoping review].pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

During active-drug treatment with octreotide, urinary 5-hydroxyindoleacetic acid (5-HIAA) excretion was reduced.

Sources[84]Published evidence snapshotClinical effects of octreotide compared to placebo in patients with gastrointestinal neuroendocrine tumours. Report on a double-blind, randomized trial.pubmed · T2
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In acromegaly, octreotide is reported to substantially reduce circulating growth hormone and/or insulin-like growth factor 1 (somatomedin C).

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Treatment response in the analyzed cohort (n=28) was 67.9% responders and 32.1% non-responders.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Symptom frequency (flushing and diarrhoea episodes) was prospectively recorded during a 1-week baseline and across the 8-week study period.

Sources[84]Published evidence snapshotClinical effects of octreotide compared to placebo in patients with gastrointestinal neuroendocrine tumours. Report on a double-blind, randomized trial.pubmed · T2
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The abstract characterizes the combination regimen (midodrine with octreotide) as commonly used in HRS-AKI when first-line or other vasoconstrictors are unavailable or impractical.

Sources[50]Published evidence snapshotMidodrine Monotherapy in Refractory Hepatorenal Syndrome-Acute Kidney Injury: A Case Report.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In acromegaly, octreotide is described as producing substantial biochemical reductions in growth hormone and/or insulin-like growth factor 1 (somatomedin C).

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Postoperative octreotide scintigraphy (octreoscan) was used for systemic evaluation, but it failed to localize a primary NET in this patient.

Sources[75]Published evidence snapshotSolitary left frontotemporal neuroendocrine metastasis mimicking a high-grade astrocytoma.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In patients with acromegaly, octreotide produces marked suppression of growth hormone and/or insulin-like growth factor 1 (somatomedin C), with normalization in many cases.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This entry reports in vitro binding affinity (Ki) for SST4; it does not specify functional activity at the receptor.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In an EBV-negative patient-derived xenograft (PDX-Li41) model, treatment with octreotide produced a statistically significant inhibition of xenograft growth.

Sources[44]Published evidence snapshotSSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is described as producing substantial suppression of GH and/or IGF-1 (somatomedin C) in acromegaly, with normalization in many cases.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The evidence base summarized in the abstract comprises three non-randomized observational studies evaluating clinical outcomes after octreotide use.

Sources[72]Published evidence snapshotEfficacy and Safety of Octreotide for Gastrointestinal Bleeding Due to Portal Hypertension in Children-A Systematic Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is indicated to lower GH and IGF-1 levels in some people with acromegaly when surgery, pituitary irradiation, and bromocriptine have not worked or cannot be used.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For patients treated with PRRT after inoperable progression following hepatic cytoreductive operation, the median overall survival reported was 97 months.

Sources[68]Published evidence snapshotpubmed-42442014pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a two-patient case series of functioning GEP-NETs (gastrinoma and VIPoma) where CE-CT was non-diagnostic, [18F]F-NOTA-octreotide PET/CT provided anatomical localization of the primary lesions.

Sources[58]Published evidence snapshotIdentification and Localization of Functioning Gastroenteropancreatic Neuroendocrine Tumors Using [18F]F-NOTA-octreotide PET/CT.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

When stratified by treatment response, the proportion with positive octreotide scintigraphy was 68.4% among responders and 77.8% among non-responders.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Post-octreotide dextrose requirements differed by octreotide route in this retrospective review, with higher dextrose administered in the infusion group than in bolus or subcutaneous groups.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a humanized mouse model (immunocompromised mice engrafted with human KCNJ11-/- SC-islets), the combination of relamorelin with octreotide is reported to act synergistically on blood glucose and to reduce excessive insulin secretion.

Sources[74]Published evidence snapshotGhrelin and relamorelin counteract hypoglycemia in mice engrafted with congenital hyperinsulinism stem cell-derived islets.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In the intention-to-treat analysis, CAM2029 increased the rate of biochemical control defined by IGF-1 ≤ULN at week 22/24 compared with placebo, with a reported risk difference and confidence interval.

Sources[38]Published evidence snapshotOctreotide Subcutaneous Depot for Acromegaly: A Randomized, Double-blind, Placebo-controlled Phase 3 Trial, ACROINNOVA 1.pubmed · T2
Human research · design must be checked

1 cited source · 1 linked study ID

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In acromegaly, octreotide (BYNFEZIA PEN) is indicated for biochemical control by reducing circulating GH and IGF-1 when standard definitive therapies (surgery/irradiation) and bromocriptine at maximally tolerated doses are inadequate or not feasible.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

The abstract describes a possible longitudinal trajectory in HI: early hyperinsulinism can be followed by impaired fasting glucose/impaired glucose tolerance and later diabetes mellitus in some individuals.

Sources[57]Published evidence snapshotA 13-Year-Old Girl with Congenital Hyperinsulinemic Hypoglycemia Due to anABCC8Mutation and Recent Onset of Diabetes Mellitus: A Case Report and Literature Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The abstract reports the sample size in terms of scans and patients and gives the cohort median age.

Sources[65]Published evidence snapshotEvaluation of [¹⁸F]AlF-NOTA-octreotide PET/CT in routine clinical use: a retrospective analysis in 288 neuroendocrine tumor patients.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

When PRRT eligibility was defined by NETTER-2 (Krenning ≥3), PET classified more patients as eligible than planar imaging performed with [111In]octreotide scintigraphy.

Sources[63]Published evidence snapshotComparison of [111In]octreotide Scintigraphy and [68Ga]DOTATOC PET in Gastroenteropancreatic Neuroendocrine Tumors: Concordance of Krenning Scores and Implications for Peptide Receptor Radionuclide Therapy Eligibility.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this randomized comparison, stool frequency control did not meaningfully differ between subcutaneous octreotide and LAR octreotide dosing groups.

Sources[29]Published evidence snapshotOctreotide Acetate Long-Acting Formulation Versus Open-Label Subcutaneous Octreotide Acetate in Malignant Carcinoid Syndromedoi · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Across EBV-positive and EBV-negative patient-derived xenograft models, the OCT-MMAE peptide-drug conjugate is reported to significantly inhibit xenograft growth.

Sources[44]Published evidence snapshotSSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Across study arms, flushing control differed by regimen: the 20-mg LAR and SC octreotide groups had the best control, while 10-mg LAR had the least effective control of flushing.

Sources[29]Published evidence snapshotOctreotide Acetate Long-Acting Formulation Versus Open-Label Subcutaneous Octreotide Acetate in Malignant Carcinoid Syndromedoi · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this real-world claims dataset, switching to OCT-LAR from LAN-ATG was associated with a 21.9% decrease in breakthrough medication claims after switching.

Sources[43]Published evidence snapshotReal-World Observational Study of Somatostatin Analogs and Rescue Medication Usage for Neuroendocrine Tumors in Canada.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study concluded that octreotide scintigraphy positivity occurred relatively frequently in patients with metastatic castration-resistant prostate cancer.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study design and inclusion window were a retrospective single-center analysis including all referrals for SSTR PET/CT during March 2023 to January 2024.

Sources[65]Published evidence snapshotEvaluation of [¹⁸F]AlF-NOTA-octreotide PET/CT in routine clinical use: a retrospective analysis in 288 neuroendocrine tumor patients.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this cohort’s liver metastases assessment, [68Ga]Ga-DOTATATE PET/CT showed lower sensitivity than [68Ga]Ga-FAP2286 (62% vs 82%).

Sources[42]Published evidence snapshotDual-tracer PET/CT and cocktail therapy with [177Lu]Lu-FAP2286 and [177Lu]Lu-DOTATATE in G3 Neuroendocrine Tumors (NET).pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study defined elevated 5-HIAA as values exceeding 45 mumol 24 h-1.

Sources[84]Published evidence snapshotClinical effects of octreotide compared to placebo in patients with gastrointestinal neuroendocrine tumours. Report on a double-blind, randomized trial.pubmed · T2
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this analysis, octreotide scan positivity did not show a statistically significant association with treatment response, with a reported P value of 1.00.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Co-administration with a permeation enhancer increased systemic exposure to octreotide in rats, as indicated by increased area under the plasma concentration–time curve (AUC), for both liquid and mini-tablet dosage forms.

Sources[71]Published evidence snapshotImpact of dosage form on the pharmacokinetics of octreotide after oral administration with permeation enhancers.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The pharmacologic effect in acromegaly includes substantial reduction of circulating growth hormone and/or IGF-I (somatomedin C).

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In this claims-based cohort, switching from OCT-LAR to LAN-ATG was associated with a 66.5% reduction in breakthrough medication claims after the switch.

Sources[43]Published evidence snapshotReal-World Observational Study of Somatostatin Analogs and Rescue Medication Usage for Neuroendocrine Tumors in Canada.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this adult-onset primary intestinal lymphangiectasia case, octreotide treatment initiation temporally coincided with gradual ascites resolution, consistent with a symptomatic improvement observed in a single patient.

Sources[52]Published evidence snapshotPrimary Intestinal Lymphangiectasia Presenting as Recurrent Chylous Ascites: A Rare Case.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

CHEMBL1680 inhibited human SSTR5 with an IC50 of 22.0 nM in a radioligand binding assay.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Sandostatin Injection is used to lower GH and IGF-1 levels in some people with acromegaly.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In CHO-K1 cells expressing human SSTR2, CHEMBL1680 inhibited forskolin-induced cAMP with EC50 = 0.03 nM (measured after 30 mins).

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

For carcinoid syndrome and VIPomas, the labeling states that effects on tumor burden and progression outcomes have not been determined for either immediate-release injection or long-acting suspension formulations.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In a database review of patients treated with PRRT after inoperable progression following HCO, the reported median progression-free survival after PRRT was 32 months.

Sources[68]Published evidence snapshotpubmed-42442014pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this spinal PMT case, the 18F-AlF-NOTA-octreotide PET/CT scan exhibited strong radiotracer uptake localized to the tumor lesion.

Sources[67]Published evidence snapshotSpinal phosphaturic mesenchymal tumor: a case report of thoracic vertebral involvement with preoperative embolization and literature review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a two-case neonatal report of mutation-associated hypoglycemia (KCNJ11/ABCC8; congenital hyperinsulinism), octreotide administration was associated with stabilization of glycemic levels, after failure of enteral/parenteral glucose infusions and lack of clinical response to diazoxide.

Sources[45]Published evidence snapshotCongenital Hyperinsulinism in Neonates: Diagnostic Challenges and Management in Two Cases With KCNJ11 and ABCC8 Mutation.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In the EBV-positive patient-derived xenograft model PDX-B13, octreotide treatment is reported to have no tumor-growth-suppressive effect.

Sources[44]Published evidence snapshotSSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is used to lower GH and IGF-1 in some people with acromegaly when surgery/irradiation/bromocriptine are not adequate or not possible.

Sources[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

3 cited sources · 3 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 3 source records.

Source-backed statement

In this reported case, disease progression occurred after initial treatment with octreotide, prompting a switch to chemotherapy (carboplatin plus etoposide).

Sources[76]Published evidence snapshotMultiple skin and subcutaneous metastasis as initial manifestation in neuroendocrine carcinoma lung: A rare case report.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

For these octreotide analogs, combining positive charge at residue 5 with higher lipophilicity (logD) is associated with greater sensitivity to phospholipid concentration in bile acid–phospholipid mixed micelles and increased micelle interaction.

Sources[80]Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is indicated to treat profuse watery diarrhea due to VIPoma-secreting tumors.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

Hospital length of stay, reported as medians, varied across octreotide administration routes in this retrospective review.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The chart review evaluated treatment intensity and resource-use endpoints as secondary outcomes: octreotide dose, dextrose administration timing around the first dose, and length of stay.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Outcome selection focused on post-octreotide hypoglycemia recurrence, measured as counts of hypoglycemic events after initiation.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Tumor-to-background ratio in liver (TBRliver) favored [68Ga]Ga-FAP2286 over [68Ga]Ga-DOTATATE in this dual-tracer PET/CT comparison.

Sources[42]Published evidence snapshotDual-tracer PET/CT and cocktail therapy with [177Lu]Lu-FAP2286 and [177Lu]Lu-DOTATATE in G3 Neuroendocrine Tumors (NET).pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study’s conclusion was that octreotide scintigraphy positivity did not show a statistically significant association with response to 177Lu-prostate-specific membrane antigen radioligand therapy.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Group sizes in the retrospective comparison were uneven, with the infusion group notably smaller than bolus or subcutaneous groups.

Sources[82]Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Comparative evidence

How the studied intervention compared with another intervention, comparator, or threshold.

8 statements
Source-backed statement

The study design included randomization, double-blinding for the LAR arms (10, 20, 30 mg every 4 weeks), and an open-label comparator arm using SC octreotide every 8 hours in carcinoid syndrome.

Sources[33]Published evidence snapshotOctreotide acetate long-acting formulation versus open-label subcutaneous octreotide acetate in malignant carcinoid syndrome.pubmed · T2
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a blinded, placebo-controlled cross-over trial, octreotide treatment was associated with significantly fewer diarrhoea and flushing episodes than placebo.

Sources[84]Published evidence snapshotClinical effects of octreotide compared to placebo in patients with gastrointestinal neuroendocrine tumours. Report on a double-blind, randomized trial.pubmed · T2
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The randomized phase 3 study used high-dose long-acting repeatable octreotide (60 mg every 4 weeks) as the control regimen.

Sources[79]Published evidence snapshotpubmed-42604001pubmed · T3
Human research · design must be checked

1 cited source · 1 linked study ID

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In the human insulinoma-derived NT-3 cell line, certain dual SSTR2/SSTR5 agonists (SMTR-002/004/005) exceeded octreotide in insulin secretion inhibition at the specified concentration.

Sources[41]Published evidence snapshotAnti-secretory and anti-proliferative actions of next-generation dual subtype 2 and 5 somatostatin receptor ligands in neuroendocrine tumor models.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The comparator in this phase 3 trial was high-dose long-acting repeatable (LAR) octreotide administered at 60 mg every 4 weeks.

Sources[79]Published evidence snapshotpubmed-42604001pubmed · T3
Human research · design must be checked

1 cited source · 1 linked study ID

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

When comparing imaging approaches, SSTR PET produced higher Krenning scores than planar imaging performed with [111In]octreotide scintigraphy, indicating stronger apparent somatostatin receptor signal on PET in this cohort.

Sources[63]Published evidence snapshotComparison of [111In]octreotide Scintigraphy and [68Ga]DOTATOC PET in Gastroenteropancreatic Neuroendocrine Tumors: Concordance of Krenning Scores and Implications for Peptide Receptor Radionuclide Therapy Eligibility.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In the pre-switch period, OCT-LAR was associated with a higher percentage of patients exceeding the above maximum recommended dose (AMRD) threshold compared with LAN-ATG, with p value = 0.008.

Sources[43]Published evidence snapshotReal-World Observational Study of Somatostatin Analogs and Rescue Medication Usage for Neuroendocrine Tumors in Canada.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The unadjusted DB proportions differed between groups: 24% (18/74) in the control group and 9% (3/33) in the octreotide group.

Sources[56]Published evidence snapshotOctreotide for prevention of delayed bleeding after endoscopic mucosal resection for large superficial non-ampullary duodenal tumors.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Mechanism

Source-backed statements about targets, pathways, and biological response.

36 statements
Source-backed statement

Octreotide is reported as a full agonist at the human somatostatin SST3 receptor, with binding affinity expressed as pKi 7.4 - 8.6.

Sources[31]Published evidence snapshotIUPHAR interactions for octreotideiuphar-interactions · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In PRRT, lutetium-177 is linked to octreotide as a radiolabeled peptide used to treat inoperable metastatic gastroenteropancreatic neuroendocrine tumors (GEPNETs).

Sources[68]Published evidence snapshotpubmed-42442014pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acts like somatostatin and more strongly inhibits growth hormone, glucagon, and insulin than somatostatin does.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

18F-AlF-NOTA-octreotide (18F-OC) is described as a targeted probe with specific binding to somatostatin receptor–expressing tumors.

Sources[60]Published evidence snapshotUptake of18F-AlF-NOTA-octreotide PET/CT in gastrointestinal stromal tumors.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

By suppressing pituitary TSH secretion, octreotide may reduce thyroid hormone signaling and lead to hypothyroidism.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The oral octreotide capsule (OOC) formulation is described as octreotide combined with transient permeability enhancer technology, implying a formulation approach to support oral delivery.

Sources[37]Published evidence snapshotOral Octreotide: A Review of Recent Clinical Trials and Practical Recommendations for Its Use in the Treatment of Patients With Acromegaly.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide in Sandostatin Injection produces somatostatin-like pharmacologic effects.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The in vitro methods described include a diffusion/transport proxy (flux through a porous cellulose dialysis membrane) and a stability assay against pancreatic enzymes.

Sources[80]Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide scintigraphy positivity was used as a surrogate indicator for neuroendocrine differentiation, and the study assessed whether that imaging marker was associated with response to 177Lu-prostate-specific membrane antigen radioligand therapy in metastatic castration-resistant prostate cancer.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

A cell-based FLIPR calcium assay using tetracycline-induced FLP-IN/T-REX 293 cells expressing an N-terminal Flag-tagged human MRGPRX2 receptor reported very low agonist potency for CHEMBL1680 (EC50 greater than 31622.78 nM).

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The abstract attributes non-diagnostic conventional imaging to tumor factors—small lesion size and heterogeneity—leading to inconclusive or false-negative scans.

Sources[58]Published evidence snapshotIdentification and Localization of Functioning Gastroenteropancreatic Neuroendocrine Tumors Using [18F]F-NOTA-octreotide PET/CT.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The biodistribution described for [¹⁸F]AlF-OC matches expected uptake in tissues that express somatostatin receptors (SSTR).

Sources[65]Published evidence snapshotEvaluation of [¹⁸F]AlF-NOTA-octreotide PET/CT in routine clinical use: a retrospective analysis in 288 neuroendocrine tumor patients.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In this report, FDG PET/CT is used to assess glucose metabolism while octreotide PET/CT is used to assess somatostatin receptor expression; the combined imaging is described as complementary for clinical evaluation.

Sources[61]Published evidence snapshotpubmed-42029102pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide served as a comparator SRL in preclinical neuroendocrine tumor cell-line assays, enabling relative assessment of novel SRLs.

Sources[41]Published evidence snapshotAnti-secretory and anti-proliferative actions of next-generation dual subtype 2 and 5 somatostatin receptor ligands in neuroendocrine tumor models.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Relative to somatostatin, octreotide has greater inhibitory potency against growth hormone, glucagon, and insulin secretion.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

Octreotide is reported as a full agonist at the human somatostatin SST2 receptor, with binding affinity expressed as pKi 8.7 - 9.9 (higher pKi indicates higher affinity).

Sources[31]Published evidence snapshotIUPHAR interactions for octreotideiuphar-interactions · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

As a somatostatin analog, octreotide produces somatostatin-like pharmacology and increases inhibitory potency against growth hormone (GH), glucagon, and insulin secretion relative to native somatostatin.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeling states octreotide suppresses pituitary TSH secretion, which can lead to hypothyroidism, supporting thyroid-function monitoring during chronic therapy.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate injection is a somatostatin analog with pharmacologic actions similar to endogenous somatostatin.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A single-protein binding assay reported binding of CHEMBL1680 to the human SST4 receptor with Ki of 66.0 nM.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study used a semi-quantitative categorization of abnormal tracer uptake (mild/moderate/severe) using liver uptake as the reference.

Sources[81]Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

A cell-based functional assay (GloSensor cAMP) in CHO-K1 cells expressing human SSTR2 reported agonist potency for CHEMBL1680, producing inhibition of forskolin-stimulated cAMP with EC50 of 0.03 nM at a 30 mins measurement time.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Based on the described findings, the authors propose further development of a combination regimen pairing relamorelin with octreotide for severe KATPHI.

Sources[74]Published evidence snapshotGhrelin and relamorelin counteract hypoglycemia in mice engrafted with congenital hyperinsulinism stem cell-derived islets.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The experimental focus was on composition-dependent effects of BAPMM, specifically varying bile salt hydroxylation state and phospholipid concentration to assess peptide–micelle interactions.

Sources[80]Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is reported as a full agonist at the human somatostatin SST5 receptor, with binding affinity expressed as pKi 7.2 - 9.5.

Sources[31]Published evidence snapshotIUPHAR interactions for octreotideiuphar-interactions · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

A single-protein binding assay reported high-affinity binding of CHEMBL1680 to the human SST2 receptor with Ki of 0.4 nM.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

SSTR signaling functions as a potent inhibitory pathway for basal secretion of pancreatic islet hormones.

Sources[64]Published evidence snapshotAmino acids partially override inhibitory effects of octreotide on islet hormone secretion in healthy individuals.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Radioligand binding data indicate low inhibitory potency of CHEMBL1680 at human SSTR4, with IC50 greater than 1000.0 nM.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

In a single-protein radioligand binding assay, CHEMBL1680 showed inhibitory binding potency at human SSTR5 with an IC50 of 22.0 nM.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

As a somatostatin analog, octreotide mimics somatostatin’s actions and is described as more potent at inhibiting secretion of growth hormone, glucagon, and insulin.

Sources[25]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Using a regression approach, the source attributes flux-rate variation primarily to an interaction term between peptide lipophilicity (logD) and the charge at residue 5 (charge5).

Sources[80]Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate can reduce pituitary thyroid-stimulating hormone (TSH) secretion.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

Octreotide has somatostatin-like pharmacodynamics, inhibiting secretion of anterior pituitary hormones (growth hormone and thyroid-stimulating hormone) and gastroenteropancreatic endocrine peptides.

Sources[36]Published evidence snapshotOctreotide. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in conditions associated with excessive peptide secretion.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

This work evaluated whether an ex vivo viability readout in patient-derived 3D tumor cultures can serve as a proxy for intrinsic pharmacologic sensitivity and whether it corresponds to established clinical predictors.

Sources[70]Published evidence snapshotEx Vivo drug sensitivity in patient-derived 3D cultures in acromegaly and its association with clinical predictors.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

SSTR2 (somatostatin receptor 2) is reported as aberrantly upregulated in various tumors, and the source states that octreotide-based molecules can be used to therapeutically target SSTR2.

Sources[53]Published evidence snapshotSSTR2 expression in EBV-positive and EBV-negative lymphomas.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide (Sandostatin) is a somatostatin analog with similar pharmacologic actions, reported to inhibit growth hormone, glucagon, and insulin more potently than somatostatin.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Pharmacokinetics

How the studied compound is absorbed, distributed, metabolized, and cleared.

18 statements
Source-backed statement

With repeated Sandostatin LAR dosing, steady-state pharmacokinetics were generally achieved by the second to third injection.

Sources[86]Published evidence snapshotSandostatin LAR (microencapsulated octreotide acetate) in acromegaly: pharmacokinetic and pharmacodynamic relationships.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Subcutaneous administration results in rapid, complete absorption of octreotide from the injection site.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Following subcutaneous administration, the reported time to peak serum concentration for octreotide is within 30 minutes.

Sources[85]Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The PK profile given indicates rapid absorption after SC administration, with a reported Cmax (5.2 ng/mL) and Tmax (0.4 hours) for a 100-mcg dose.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For a three minute intravenous infusion, octreotide reaches peak serum concentrations within four minutes.

Sources[85]Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Subcutaneous administration results in rapid and complete absorption of octreotide from the injection site.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide is described as rapidly distributing with predominant plasma distribution and 65% plasma protein binding.

Sources[85]Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

CAM2029 is formulated with FluidCrystal technology, which the source states increases the bioavailability of octreotide (more drug becomes available systemically).

Sources[38]Published evidence snapshotOctreotide Subcutaneous Depot for Acromegaly: A Randomized, Double-blind, Placebo-controlled Phase 3 Trial, ACROINNOVA 1.pubmed · T2
Human research · design must be checked

1 cited source · 1 linked study ID

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide shows an apparent plasma elimination half-life in the range of 1.7 to 1.9 hours.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

These pharmacokinetic values are reported for subcutaneous dosing and depend on the assay and study conditions; they do not directly predict clinical effect.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A cell-free assay measuring stability in human plasma reported a half-life (T1/2) of 1.5 hr for CHEMBL1680.

Sources[5]Published evidence snapshotChEMBL activities for CHEMBL1680chembl-activities · T6
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Following subcutaneous dosing, the source reports that about 32% of octreotide is recovered in urine as unchanged drug.

Sources[85]Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

With the immediate-release formulation given subcutaneously, octreotide shows rapid absorption with reported Cmax 5.2 ng/mL after a 100-mcg dose at 0.4 hours (Tmax).

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

After a 100-mcg subcutaneous dose, peak blood levels were 5.2 ng/mL at 0.4 hours.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

With immediate-release octreotide acetate injection given subcutaneously, systemic exposure peaks rapidly; for a 100 mcg dose, Cmax is 5.2 ng/mL at 0.4 hours.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For immediate-release octreotide acetate injection, the text reports a peak concentration (Cmax) of 5.2 ng/mL after a 100-mcg subcutaneous dose, occurring at 0.4 hours (Tmax).

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Double-blind single-dose clinical studies in acromegaly evaluated 10, 20, and 30 mg Sandostatin LAR to characterize its pharmacokinetic profile.

Sources[86]Published evidence snapshotSandostatin LAR (microencapsulated octreotide acetate) in acromegaly: pharmacokinetic and pharmacodynamic relationships.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Relative to endogenous somatostatin (minutes), octreotide has a longer apparent plasma elimination half-life (hours).

Sources[21]Published evidence snapshotRx ONLYdailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Safety findings

Observed or labeled risks, adverse effects, and safety signals.

18 statements
Source-backed statement

The source states a mechanistic safety concern: octreotide may reduce gallbladder motility and bile secretion, predisposing to biliary abnormalities (e.g., sludge).

Sources[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

3 cited sources · 3 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 3 source records.

Source-backed statement

By decreasing gallbladder motility and bile secretion, octreotide depot therapy may predispose to biliary sludge or other gallbladder abnormalities.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Clinical-trial safety data in mainly acromegaly/psoriasis populations reported frequent biliary tract abnormalities during chronic octreotide acetate injection therapy, with specific proportions for gallstones, sludge, and biliary duct dilatation.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Immunogenicity assessment in an open-label study found no detectable anti-octreotide antibodies (per the assay used) among 149 assessed patients during 13 months of MYCAPSSA treatment.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

An overdosage statement reports specific adverse effects (hypoglycemia, flushing, dizziness, nausea) associated with 2.5 mg (2,500 mcg) subcutaneous octreotide acetate injection.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

By altering counter-regulatory hormones (including insulin and glucagon), octreotide therapy may produce hypoglycemia or hyperglycemia; the label provides frequencies in acromegaly patients.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Clinical trials cited in labeling report a high incidence of biliary tract abnormalities during Sandostatin Injection therapy, with specific proportions for gallstones, sludge without stones, and biliary duct dilatation.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A stated adverse physiology mechanism is reduced gallbladder contractility and bile secretion, which can predispose to gallbladder abnormalities or sludge.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In acromegaly populations treated with octreotide acetate injection or the long-acting injectable suspension, reported glucose disturbances included hypoglycemia (~2%) and hyperglycemia (~15%).

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Clinical trial safety data for MYCAPSSA include reported glucose-related adverse reactions: hyperglycemia/increased blood glucose, hypoglycemia, and diabetes mellitus, with stated percentages.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The warning section quantifies biliary tract abnormalities seen in trials (primarily in acromegaly or psoriasis) during octreotide acetate therapy, including gallstones, sludge, and duct dilatation.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide therapy (MYCAPSSA) can change endocrine counter-regulation involving insulin, glucagon, and GH, predisposing to dysglycemia including hypoglycemia, hyperglycemia, and diabetes mellitus.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

TSH suppression is described as a pharmacodynamic effect of octreotide, with possible clinical consequence of hypothyroidism.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Cardiac-related adverse reactions reported in MYCAPSSA trials include bradycardia, conduction abnormalities, and arrhythmias/tachycardia with stated incidence percentages.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

By altering counter-regulatory hormones (insulin, glucagon, and growth hormone), octreotide may dysregulate glycemia, leading to hypoglycemia or hyperglycemia.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide (Sandostatin Injection) is reported to inhibit gallbladder contractility and decrease bile secretion, which may contribute to biliary abnormalities such as sludge.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Immunogenicity testing in an open-label MYCAPSSA study found no detectable anti-octreotide peptide antibodies among 149 assessed patients over 13 months.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

MYCAPSSA clinical trial safety reporting includes thyroid-related adverse reactions (hypothyroidism, increased thyroid-stimulating hormone, and decreased free thyroxine), each at 1%.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Contraindications

Circumstances in which a specific product label says it should not be used.

9 statements
Source-backed statement

The contraindication is hypersensitivity to octreotide acetate or excipients/components of the product.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Do not take MYCAPSSA if you are hypersensitive to octreotide or its ingredients; severe allergic reactions (including anaphylactic shock) have been reported with octreotide.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled contraindication is hypersensitivity to Sandostatin Injection or its components.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Contraindication: prior hypersensitivity to the active peptide (octreotide) or excipients precludes use.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled contraindication for MYCAPSSA is hypersensitivity to the active peptide (octreotide) or excipients in the product.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The contraindication is stated as hypersensitivity; the section also notes reported anaphylactoid reactions with octreotide.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled contraindication is allergy/hypersensitivity to the active peptide (octreotide) or excipients in MYCAPSSA, reflecting risk of serious allergic reactions.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A labeled contraindication is hypersensitivity to octreotide or formulation components; severe immediate hypersensitivity reactions have been reported with octreotide exposure.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeling states SANDOSTATIN LAR DEPOT must not be administered by IV or subcutaneous routes.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Interactions

Source-backed product and drug interaction statements.

5 statements
Source-backed statement

A drug–drug interaction finding reported is reduced oral bioavailability of MYCAPSSA when co-administered with the proton pump inhibitor esomeprazole, consistent with pH-dependent absorption effects.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Competitive binding at somatostatin receptors is stated as the mechanism for potential reduction in lutetium Lu 177 dotatate efficacy when used with octreotide.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A drug–drug interaction is described in which octreotide injection can decrease cyclosporine blood concentrations, with potential clinical consequence of transplant rejection.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A potential drug interaction is reduced cyclosporine exposure when co-administered with octreotide acetate injection, with possible clinical consequence of transplant rejection.

Sources[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In Total Parenteral Nutrition (TPN) solutions, octreotide acetate injection is incompatible due to formation of a glycosylated octreotide conjugate, which may lower product efficacy.

Sources[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Regulatory status

Product-, indication-, and jurisdiction-specific regulatory records.

37 statements
Source-backed statement

This labeled indication is for diarrhea control in VIPoma-secreting tumors; it does not claim tumor reduction.

Sources[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication for oral octreotide (MYCAPSSA) is long-term maintenance therapy in acromegaly, specifically for patients already shown to respond to and tolerate prior somatostatin analog therapy (octreotide or lanreotide).

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 2 source records.

Source-backed statement

The labeled indication includes treatment of profuse watery diarrhea associated with vasoactive intestinal peptide tumor (VIPoma) secretion.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For vasoactive intestinal peptide–secreting tumors (VIPomas), octreotide acetate injection is indicated to treat the associated profuse watery diarrhea.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

8 cited sources · 8 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

10 cited passages across 8 source records.

Source-backed statement

This indication is conditional on prior response and tolerability to Sandostatin Injection; it does not specify a disease by itself in this sentence.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For carcinoid syndrome and VIPomas, it is not known whether octreotide affects tumor size, growth rate, or metastases.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication for the long-acting injectable suspension specifies use in patients with demonstrated effectiveness and tolerability on initial octreotide acetate injection.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

MYCAPSSA is used as long-term maintenance treatment for acromegaly in people who responded to and tolerated octreotide or lanreotide.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes acromegaly requiring biochemical reduction of GH and IGF‑I when standard interventions (resection, irradiation, bromocriptine) are ineffective or not feasible.

Sources[21]Published evidence snapshotRx ONLYdailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For acromegaly, octreotide acetate for injectable suspension is indicated for long-term maintenance in patients with inadequate response to surgery and/or radiotherapy or when those options are unsuitable.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

MYCAPSSA is used as long-term maintenance treatment for acromegaly in patients who responded to and tolerated octreotide or lanreotide.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This section states intended use and a treatment goal (biochemical targets) but does not quantify expected response for any specific regimen.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For acromegaly, octreotide acetate long-acting injectable suspension is indicated as long-term maintenance when surgery and/or radiotherapy is inadequate or not feasible.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For carcinoid syndrome and VIPoma indications, the labeling states that antitumor outcomes (tumor size, growth kinetics, metastasis development) have not been determined for octreotide acetate injection or the injectable suspension.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

This indication is limited to patients whose initial treatment with octreotide acetate injection was effective and tolerated; it does not state benefit in injection-naïve patients.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeling states that antitumor effects (tumor size, growth rate, metastasis development) have not been determined for octreotide acetate injection or the long-acting injectable suspension in carcinoid syndrome and VIPomas.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

For acromegaly, Sandostatin Injection is indicated to reduce circulating GH and IGF-1 when standard interventions (surgical resection, pituitary irradiation, maximally tolerated bromocriptine) are inadequate or not feasible.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes biochemical reduction of GH and IGF-1 in acromegaly when surgical resection, pituitary irradiation, and maximally tolerated bromocriptine mesylate are not effective or not feasible.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For VIPomas (VIP-secreting tumors), octreotide acetate for injectable suspension is indicated for long-term treatment of profuse watery diarrhea.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

4 cited passages across 2 source records.

Source-backed statement

For acromegaly, SANDOSTATIN LAR DEPOT is labeled for long-term maintenance when definitive local therapies (surgery/radiotherapy) fail or cannot be used.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes management of VIPoma-associated secretory diarrhea.

Sources[21]Published evidence snapshotRx ONLYdailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes biochemical reduction of GH and IGF-1 in acromegaly patients who have not responded adequately to, or cannot receive, surgery, pituitary irradiation, and bromocriptine mesylate at maximally tolerated doses.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For metastatic carcinoid tumors, octreotide acetate injection is an indicated symptomatic treatment for severe diarrhea and flushing episodes.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

8 cited sources · 8 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

11 cited passages across 8 source records.

Source-backed statement

For VIP-secreting tumors, octreotide acetate injection is indicated to treat the associated profuse watery diarrhea.

Sources[16]Published evidence snapshotRx OnlyPrescribing Informationdailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

A labeled limitation notes that antitumor outcomes (tumor size, growth rate, metastases) have not been determined for octreotide (immediate-release or LAR) in carcinoid syndrome and VIPomas.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes biochemical reduction of growth hormone (GH) and insulin-like growth factor-1 (IGF-1; somatomedin C) in acromegaly when standard interventions (resection, irradiation, bromocriptine at maximally tolerated doses) are insufficient or not feasible.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For VIPoma-associated secretory diarrhea, Sandostatin Injection is indicated to treat profuse watery diarrhea.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes symptomatic treatment of severe diarrhea and flushing episodes associated with metastatic carcinoid tumors.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication includes treatment of profuse watery diarrhea associated with vasoactive intestinal peptide tumor (VIPoma) secretion.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For metastatic carcinoid tumors, octreotide acetate for injectable suspension is indicated for long-term management of severe diarrhea and flushing episodes.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

4 cited passages across 2 source records.

Source-backed statement

Octreotide injection is indicated to lower GH and IGF‑I in acromegaly when surgery, pituitary irradiation, and maximally tolerated bromocriptine are inadequate or not possible.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled indication for the long-acting injectable suspension requires prior demonstration that immediate-release octreotide acetate injection was effective and tolerated.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

4 cited passages across 2 source records.

Source-backed statement

This indication specifies use of the long-acting depot formulation only after effectiveness and tolerability are demonstrated with Sandostatin Injection.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled use includes maintenance therapy for acromegaly in patients with inadequate response to, or inability to undergo, surgery and/or radiotherapy.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeling states that tumor-related outcomes (size, growth rate, metastasis development) have not been determined for these conditions.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

MYCAPSSA (oral octreotide) has an approved indication for maintenance therapy in acromegaly after prior response and tolerability to somatostatin analog therapy (octreotide or lanreotide).

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This statement describes the indicated acromegaly use context (post-surgery/radiotherapy inadequate response or not feasible) but does not provide response rates here.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Administration

Product-specific route, timing, formulation, and use instructions—not universal dosing advice.

15 statements
Source-backed statement

IV administration options include dilution (50–200 mL) for infusion over 15–30 minutes, or IV push administration over 3 minutes.

Sources[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

The labeled routes of administration for Sandostatin Injection include subcutaneous injection and intravenous administration.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

The labeled subcutaneous injection sites for BYNFEZIA PEN include abdomen, anterior mid-thigh, and posterior/lateral upper arm, supporting site selection for routine administration.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

Initial SC dosing in acromegaly begins at 50 mcg three times daily, with subsequent titration based on biochemical markers.

Sources[18]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Administration instructions specify oral dosing under fasting conditions to support absorption, and the delayed-release capsule should remain intact (no crushing/chewing) to preserve its release characteristics.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 1 source record.

Source-backed statement

The dosing instructions specify two parenteral routes (SC or IV), with SC described as the usual route when using octreotide acetate for symptom control.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Administration instructions specify fasting administration with water and intact swallowing to preserve the delayed-release capsule performance.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate for injectable suspension is given as a gluteal IM injection every 4 weeks and should not be given IV or under the skin.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The depot formulation is administered IM (gluteal) on a 4-week schedule; IV and subcutaneous routes are contraindicated for administration.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The long-acting injectable suspension formulation is administered via intramuscular injection into the gluteal region on a 4-week dosing interval.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The product’s dosage forms/strengths are single-dose vials containing octreotide acetate injection at concentrations of 100 mcg per mL and 500 mcg per mL.

Sources[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The labeled route/site and schedule for SANDOSTATIN LAR DEPOT is intramuscular (gluteal) administration at 4-week intervals.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial carcinoid syndrome dosing is subcutaneous, divided 2–4 times daily, totaling 100–600 mcg/day for the first 2 weeks.

Sources[18]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The product labeling permits parenteral administration by either subcutaneous (SC) injection or intravenous (IV) administration.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[25]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

The product is labeled for intramuscular administration in the gluteal region on a 4-week dosing interval, with explicit instructions to avoid intravenous or subcutaneous administration.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Dose records

Product- and indication-specific dose statements preserved separately to prevent unsafe generalization.

45 statements
Source-backed statement

The labeling recommends initiating octreotide acetate for acromegaly at 50 mcg subcutaneously three times daily before titration based on GH or IGF-1.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial carcinoid dosing guidance specifies 100–600 mcg/day SC, split into 2–4 doses, for the first 2 weeks (mean 300 mcg/day).

Sources[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Recommended starting regimen for oral octreotide (MYCAPSSA) is 40 mg/day split into 20 mg BID dosing.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

Initial carcinoid-tumor dosing guidance recommends 100–600 mcg/day of octreotide acetate injection subcutaneously, split into 2–4 doses, during the first 2 weeks.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

If a patient has established liver cirrhosis, start octreotide acetate for injectable suspension at 10 mg every 4 weeks.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For carcinoid tumors (first 2 weeks), the dose is 100 to 600 mcg/day under the skin in 2 to 4 divided doses.

Sources[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For cirrhotic patients, labeling recommends a reduced starting dose regimen of 10 mg every 4 weeks.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial carcinoid dosing guidance specifies 100–600 mcg/day given subcutaneously in 2–4 divided doses for the first 2 weeks (mean 300 mcg/day).

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This section provides a specific starting dose for ESRD; subsequent titration is based on IGF-1, signs/symptoms, and tolerability.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial dosing guidance for VIPomas recommends subcutaneous octreotide acetate injection 200–300 mcg/day in 2–4 divided doses during the initial 2 weeks; a wider range of 150–750 mcg is noted for symptom control.

Sources[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In end-stage renal disease, start MYCAPSSA at 20 mg once daily by mouth.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The dosage form is a prefilled pen delivering a clear, colorless octreotide acetate solution at 2,500 mcg/mL, totaling 7,000 mcg per 2.8 mL pen.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For renal failure requiring dialysis, labeling recommends initiating octreotide acetate for injectable suspension at 10 mg once every 4 weeks.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

Initial (first 2 weeks) dosing guidance for carcinoid tumors recommends subcutaneous octreotide acetate injection totaling 100–600 mcg/day in 2–4 divided doses; mean daily dose is 300 mcg.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

In acromegaly, octreotide acetate injection is initiated at 50 mcg SC three times daily before titration based on GH or IGF-1 levels.

Sources[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

The labeled initial dosing for dialysis-dependent renal failure is 10 mg of SANDOSTATIN LAR DEPOT administered every 4 weeks.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For metastatic carcinoid tumor symptoms, the first 2 weeks dose range is 100 to 600 mcg/day given subcutaneously in 2 to 4 divided doses.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial titration in acromegaly begins with subcutaneous octreotide 50 mcg TID, with subsequent dose adjustments guided by biochemical monitoring elsewhere in the regimen.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Dose ceiling: MYCAPSSA is not recommended above 80 mg/day per labeling.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For VIPomas (first 2 weeks), the recommended dose is 200 to 300 mcg/day under the skin in 2 to 4 divided doses.

Sources[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In acromegaly, the labeled initial regimen is 50 mcg subcutaneously three times daily.

Sources[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

3 cited sources · 3 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 3 source records.

Source-backed statement

This section specifies a cirrhosis starting dose; subsequent titration guidance is not included in this section.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial treatment dosing guidance for carcinoid tumors specifies a subcutaneous total daily dose range and divided dosing frequency over the first 2 weeks.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial dosing guidance for acromegaly specifies subcutaneous octreotide acetate injection at 50 mcg three times daily.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

For acromegaly patients transitioning from immediate-release octreotide acetate injection, the label recommends initiating the long-acting suspension at 20 mg IM intragluteally every 4 weeks for 3 months before titration.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This section states biochemical targets used to guide titration/monitoring; it does not provide evidence that these targets are always achieved.

Sources[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

If already on Sandostatin Injection for acromegaly, the label describes switching to Sandostatin LAR Depot 20 mg IM every 4 weeks for 3 months.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For acromegaly, the recommended starting dose is 50 mcg under the skin 3 times a day.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 2 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

For VIPomas, the initial 2 weeks recommend 200 to 300 mcg/day under the skin in 2 to 4 divided doses (range 150 to 750 mcg) to control symptoms.

Sources[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial VIPoma dosing recommends SC dosing divided 2–4 times daily totaling 200–300 mcg/day (range 150–750 mcg) during the first 2 weeks for symptom control.

Sources[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Dose escalation for MYCAPSSA has an upper recommended limit of 80 mg per day; titration beyond this is not recommended per the dosing section.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In acromegaly patients already on octreotide acetate injection, the recommended switch is 20 mg IM (intragluteal) every 4 weeks for 3 months.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For carcinoid tumors, during the first 2 weeks the recommended total daily dose is 100–600 mcg/day in 2–4 under-the-skin doses.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial dosing guidance for acromegaly is 50 mcg administered subcutaneously three times per day.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 1 source record.

Source-backed statement

For acromegaly, start BYNFEZIA PEN at 50 mcg under the skin 3 times daily.

Sources[8]Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Labeling specifies a lower starting dose of oral octreotide (MYCAPSSA) in ESRD, with subsequent individualized maintenance dosing guided by IGF-1 and clinical response/tolerability.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Titration is guided by biochemical control (IGF-1) and clinical status, using stepwise 20 mg/day increases.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial therapy for carcinoid tumors uses subcutaneous octreotide acetate injection at 100–600 mcg/day for the first 2 weeks, split into 2 to 4 doses.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

5 cited sources · 5 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

5 cited passages across 5 source records.

Source-backed statement

The labeled capsule strength for oral delayed-release octreotide (MYCAPSSA) is 20 mg of octreotide content, supplied as the acetate salt.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In VIPoma-associated watery diarrhea, recommended initial dosing for symptom control over the first 2 weeks is 200–300 mcg/day subcutaneously in 2–4 divided doses.

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This statement applies to renal failure requiring dialysis; other renal impairment starting dose is addressed separately in the same section.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For vasoactive intestinal peptide tumors (VIPomas), the recommended starting regimen over the initial 2 weeks is subcutaneous octreotide 200–300 mcg/day divided into 2 to 4 doses.

Sources[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Initial VIPoma dosing recommendations specify 200–300 mcg/day SC divided into 2–4 doses for the initial 2 weeks (range 150–750 mcg) for symptom control.

Sources[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In acromegaly dosing, octreotide acetate is initiated at 50 mcg SC three times daily before titration based on GH/IGF-1.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

For acromegaly dosing initiation, octreotide acetate injection is started at 50 mcg SC three times daily.

Sources[10]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[23]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[27]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

5 cited sources · 5 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

5 cited passages across 5 source records.

Studied populations

Who was represented in a study, label, or registry record.

4 statements
Source-backed statement

Dose initiation in renal failure requiring dialysis is reduced: octreotide acetate long-acting suspension should start at 10 mg administered every 4 weeks.

Sources[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This applies specifically to renal failure requiring dialysis and refers to starting dose.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Renal special population dosing: ESRD patients start at a lower initial oral dose (20 mg QD), with later adjustment based on response/tolerability.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

This applies to established cirrhosis and addresses only the starting dose.

Sources[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Identity

Ingredient, molecule, and product identity statements.

44 statements
Source-backed statement

The injection is supplied in sterile 1 mL ampuls with three labeled strengths: 50 mcg, 100 mcg, or 500 mcg octreotide (as acetate).

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The source characterizes congenital hyperinsulinism (HI) as genetically heterogeneous, with underlying disorders that disrupt regulation of insulin secretion.

Sources[57]Published evidence snapshotA 13-Year-Old Girl with Congenital Hyperinsulinemic Hypoglycemia Due to anABCC8Mutation and Recent Onset of Diabetes Mellitus: A Case Report and Literature Review.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is an acetate-salt, cyclic octapeptide drug product supplied as a sterile solution intended for parenteral administration (deep subcutaneous/intrafat or intravenous).

Sources[19]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate injection is formulated as a cyclic octapeptide (octreotide acetate salt) intended for parenteral administration by deep subcutaneous or intravenous injection.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The case included germline genetic testing identifying a VHL p.Asp126Asn variant.

Sources[61]Published evidence snapshotpubmed-42029102pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

CAM2029 is an octreotide formulation designed as a subcutaneous depot (a long-acting injectable form placed under the skin).

Sources[38]Published evidence snapshotOctreotide Subcutaneous Depot for Acromegaly: A Randomized, Double-blind, Placebo-controlled Phase 3 Trial, ACROINNOVA 1.pubmed · T2
Human research · design must be checked

1 cited source · 1 linked study ID

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The abstract states the creation of OCT-MMAE, a peptide-drug conjugate linking octreotide to monomethyl auristatin E.

Sources[44]Published evidence snapshotSSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is referenced as one of the long-acting somatostatin analogs considered in studies of gastroenteropancreatic neuroendocrine neoplasm (GEP-NEN) management.

Sources[78]Published evidence snapshotEditorial: Toward Prognostic Precision in the Management of Gastroenteropancreatic Neuroendocrine Neoplasms.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide Acetate Injection comes as a clear, single-dose vial: 50, 100, or 500 mcg per mL (as acetate).

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The IUPHAR entry classifies [<sup>67</sup>Ga]NODAGA-[Tyr<sup>3</sup>]octreotide (Ligand ID 5628) as a peptide ligand.

Sources[32]Published evidence snapshot[<sup>67</sup>Ga]NODAGA-[Tyr<sup>3</sup>]octreotideiuphar-ligand · T6
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is formulated as a cyclic octapeptide (octreotide, acetate salt) in a sterile solution designed for parenteral administration by deep subcutaneous or intravenous injection.

Sources[7]Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[16]Published evidence snapshotRx OnlyPrescribing Informationdailymed · T1[17]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[18]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1[28]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

6 cited sources · 6 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

6 cited passages across 6 source records.

Source-backed statement

Octreotide acetate has a microencapsulated long-acting (LAR) formulation intended to enable monthly intramuscular administration.

Sources[33]Published evidence snapshotOctreotide acetate long-acting formulation versus open-label subcutaneous octreotide acetate in malignant carcinoid syndrome.pubmed · T2
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The dosage forms and strengths include clear-solution single-dose vials containing octreotide (as acetate) at concentrations of 100 mcg/mL or 500 mcg/mL.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate is a cyclic octapeptide (as an acetate salt) supplied as a sterile injectable solution intended for deep subcutaneous or intravenous administration.

Sources[11]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide is described as a water-soluble cyclic octapeptide.

Sources[80]Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.pubmed · T3
Animal / laboratory evidence

1 cited source · Study independence not established

Animal or laboratory findings do not establish benefit or safety in people.

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The dosage forms/strengths list octreotide (as acetate) injection as a clear solution in multi-dose vials at concentrations of 200 mcg/mL and 1000 mcg/mL.

Sources[9]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate injection contains the peptide octreotide (as the acetate salt) formulated as a buffered acetic acid sterile solution for SC or IV administration.

Sources[21]Published evidence snapshotRx ONLYdailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

In 68Ga-DOTATOC PET-CT, the imaging agent is octreotide (DOTA-D-Phe-Tyr-octreotide) labelled with gallium-68 to enable PET/CT detection.

Sources[47]Published evidence snapshotPulmonary neuroendocrine tumour-associated ectopic Cushing's syndrome: diagnostic challenges and multidisciplinary management.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is formulated as the acetate salt in a sterile solution and is intended for parenteral dosing by deep subcutaneous (intrafat) or intravenous injection.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide in Sandostatin Injection is a cyclic octapeptide provided as the acetate salt in a buffered lactic acid solution intended for deep subcutaneous or intravenous administration.

Sources[12]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate is categorized as a somatostatin receptor ligand used in acromegaly pharmacotherapy.

Sources[55]Published evidence snapshotDevelopments in Pharmacotherapy for Acromegaly: Current and Emerging Approaches.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is categorized as a somatostatin analog and is listed among primary treatments for autosomal dominant polycystic kidney disease (ADPKD) or polycystic liver disease (PLD).

Sources[69]Published evidence snapshotComparative Efficacy and Safety of Octreotide, Lanreotide, and Pasireotide in ADPKD and PLD: A Network Meta-analysis with Real-world Evidence from the FAERS Database.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is identified here as a somatostatin analogue (a drug that mimics somatostatin signaling).

Sources[83]Published evidence snapshotDifferential Somatostatin Sensitivity of Corticotropic and Somatotropic Responses Following Amino Acid Infusion.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide subcutaneous (SC) depot is categorized as a somatostatin receptor ligand used in acromegaly pharmacotherapy.

Sources[55]Published evidence snapshotDevelopments in Pharmacotherapy for Acromegaly: Current and Emerging Approaches.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is described as an 8-amino-acid cyclic peptide (a small cyclic peptide drug).

Sources[48]Published evidence snapshotEffect of octreotide-deoxycholate hydrophobic ion pairing solid dispersions on intestinal permeability to enhance octreotide absorption via increased lipophilicity and ASBT-mediated transport.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is a somatostatin analogue (a compound designed to mimic somatostatin’s actions).

Sources[36]Published evidence snapshotOctreotide. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in conditions associated with excessive peptide secretion.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Within the study’s treatment taxonomy for malignant bowel obstruction, octreotide was specified as a medical management option.

Sources[49]Published evidence snapshotMedical Versus Surgical/Endoscopic Management of Malignant Bowel Obstruction in Patients With End-Stage Gynecologic Cancer: A 12-Year Single-Center Experience.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

DOTATATE here is explicitly defined as [177Lu]Lu(lutetium)-(DOTA0, Tyr3) octreotide, i.e., an octreotide-based radioligand.

Sources[42]Published evidence snapshotDual-tracer PET/CT and cocktail therapy with [177Lu]Lu-FAP2286 and [177Lu]Lu-DOTATATE in G3 Neuroendocrine Tumors (NET).pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection comes as a clear, single-dose vial at 100 mcg/mL.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The active drug substance in MYCAPSSA is octreotide acetate, a somatostatin analog formulated as delayed-release oral capsules.

Sources[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

The molecular formula given for octreotide specifies its elemental composition as C49H66N10O10S2.

Sources[6]Published evidence snapshotOCTREOTIDEchembl-molecule · T6
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The dosage form/strength specified is a clear single-dose vial solution containing octreotide (as acetate) at 100 mcg/mL.

Sources[20]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide is a synthetic somatostatin analogue composed of 8 amino acids.

Sources[85]Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide was part of a set of additional cyclic peptides used for comparative validation of a graph-theoretic framework applied to cyclic peptide molecular graphs.

Sources[77]Published evidence snapshotStructural control and resilience in the oxytocin molecular graph: A graph-theoretic framework for critical atom and bond identification with comparative validation across cyclic peptides.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Formulation/strength: MYCAPSSA is an oral delayed-release capsule delivering 20 mg of the peptide octreotide in the acetate salt form.

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate in MYCAPSSA is classified as a somatostatin analog (a peptide drug that mimics somatostatin-like pharmacology).

Sources[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1[15]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

2 cited sources · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

2 cited passages across 2 source records.

Source-backed statement

Oral octreotide is categorized as a somatostatin receptor ligand used in acromegaly pharmacotherapy.

Sources[55]Published evidence snapshotDevelopments in Pharmacotherapy for Acromegaly: Current and Emerging Approaches.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is a cyclic octapeptide presented as an acetate salt, i.e., an 8-residue peptide with a cyclic structure formulated with acetate.

Sources[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[24]Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1[26]Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
Regulatory record

3 cited sources · 3 regulatory records

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

3 cited passages across 3 source records.

Source-backed statement

The source notes ambiguity in stereochemical representation for octreotide; the displayed structure omits stereochemistry, which can lead to differences versus other chemical resources.

Sources[30]Published evidence snapshotIUPHAR ligand commentaryiuphar-comments · T6
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

The study administered a radiolabeled octreotide analogue, 177Lu-DOTA-TATE, as the PRRT compound.

Sources[73]Published evidence snapshotAnalysis of outcome in patients with different primary localisation of neuroendocrine tumors after PRRT. 10 years single institution experience.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide long-acting release (LAR) is categorized as a somatostatin receptor ligand used in acromegaly pharmacotherapy.

Sources[55]Published evidence snapshotDevelopments in Pharmacotherapy for Acromegaly: Current and Emerging Approaches.pubmed · T3
Human research · design must be checked

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide is a cyclic peptide made of eight amino acids with long-acting somatostatin-like pharmacologic activity.

Sources[35]Published evidence snapshotDebut of a somatostatin analog: octreotide in review.pubmed · T3
Molecular / pharmacology evidence

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Source-backed statement

Octreotide acetate injection is a cyclic octapeptide solution given by deep subcutaneous or intravenous injection.

Sources[14]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Source-backed statement

Octreotide acetate (a somatostatin analog) is described as a cyclic octapeptide provided as a sterile injectable solution (acetate salt).

Sources[25]Published evidence snapshotOctreotide Acetate Injectiondailymed · T1
Regulatory record

1 cited source · 1 regulatory record

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record.

Additional research & classification gaps

39 archived statements are kept separate from drug-effect findings. Media studies, economic models, methods, and records with unresolved scope are not used as medical-effect evidence.

Inspect contextual research (39)
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In NT-3 3D spheroid cultures, SMTR-002’s antisecretory effect on insulin was reported as comparable to octreotide, indicating similar magnitude in that model.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In a nationwide survey assessing HRS-AKI management practices, respondents reported first-line vasoconstrictor regimen preferences; midodrine/octreotide was selected by 44% of providers, while terlipressin was selected by 49%.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Across the peptide set, bile salt hydroxylation state matters: dihydroxy BAPMM produces stronger peptide–micelle interactions than trihydroxy BAPMM.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The stated objective was to evaluate an association between postprocedural octreotide exposure and delayed bleeding following duodenal EMR in large superficial non-ampullary duodenal tumors.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Co-infusion of octreotide attenuated amino-acid–stimulated islet hormone responses, leaving 49% of the glucagon response, 43% of the insulin response, and 78% of the C‑peptide response compared with amino acids alone.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The review defined its primary endpoint as resolution of crisis symptoms.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

When residue 5 carries a negative charge, the octreotide analogs show reduced sensitivity to phospholipid concentration changes in the BAPMM system.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In this report, combining 18 F-FDG PET/CT (glucose metabolism) with 18 F-octreotide PET/CT (somatostatin receptor expression) yielded complementary imaging information for VHL-mutated pheochromocytoma.

Research context only—not evidence of a treatment effect.

  • pubmed-42029102
    This "dual-tracer" strategy provided complementary information on glucose metabolism and somatostatin receptor expression, facilitating prognostic stratification and therapeutic decision-making in VHL-mutated pheochromocytoma.
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Transcriptomic and protein analyses in the EBV-negative PDX-Li41 model found heterogeneous regulation of cell-cycle-related genes with pathway-level shifts: DNA replication pathways were upregulated, while cell-signaling and neurotransmitter-release pathways were downregulated after octreotide treatment.

Research context only—not evidence of a treatment effect.

  • SSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.
    In the EBV-negative PDX-Li41 model, treatment with the SSTR2 agonist octreotide (OCT) significantly inhibited xenograft growth and showed additive effects with chemotherapy; transcriptomic and protein analyses revealed heterogeneous regulation of cell-cycle-related genes, upregulation of DNA replication pathways, downregulation of cell-signaling and neurotransmitter-release pathways,
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Amino acids act as strong secretagogues for glucagon release.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In carcinoid syndrome, subcutaneous octreotide acetate is stated to effectively relieve two hallmark symptoms: diarrhea and flushing.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In a Caco-2 intestinal epithelial cell model, complexing octreotide with stearic acid-functionalised mesoporous silica increased measured trans-epithelial transport versus unformulated octreotide.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Using immunohistochemistry in a retrospective set of lymphoma cases, the study reports SSTR2 positivity in 43% (20/47) of EBV-positive classic Hodgkin lymphoma and none (0/12) of EBV-negative classic Hodgkin lymphoma.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In the Caco-2 permeability assay, adding the permeation enhancer SNAC to octreotide produced a measured transport value of 2.59 ± 0.38%.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In the EBV-negative PDX-Li41 xenograft model, transcriptomic/protein analyses reported reduced expression of specific regulators (CDK6, NF-κB, E2F1, CDK2) and BIRC5 following octreotide treatment.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Among EBV-negative follicular lymphoma cases in this series, SSTR2 expression by immunohistochemistry is reported in 17% (5/29).

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The octreotide–monomethyl auristatin E conjugate (OCT-MMAE) is reported to internalize into cells efficiently (no assay details provided in the abstract).

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Relative to glucose, amino acids are weaker stimuli for insulin secretion.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The abstract states that SC octreotide acetate is effective for relieving two key carcinoid syndrome symptoms: diarrhea and flushing.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

This source lists SMS995 as an alternate identifier/name for octreotide.

Research context only—not evidence of a treatment effect.

  • OCTREOTIDE
    Octreotida; Octreotide; SMS 201-995; SMS-201-995; SMS-995; SMS995
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

18F-AlF-NOTA-octreotide is described as a fluorinated ligand that targets somatostatin receptors for PET imaging.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

This source lists alternate names (synonyms) for octreotide, including Octreotida.

Research context only—not evidence of a treatment effect.

  • OCTREOTIDE
    Octreotida; Octreotide; SMS 201-995; SMS-201-995; SMS-995; SMS995
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Octreotide subcutaneous depot is called CAM2029.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The source lists SMS 201-995 as an alternate name used for octreotide.

Research context only—not evidence of a treatment effect.

  • OCTREOTIDE
    Octreotida; Octreotide; SMS 201-995; SMS-201-995; SMS-995; SMS995
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

ChEMBL lists OCTREOTIDE as the preferred name for this molecule entry.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Octreotide is described as a somatostatin mimetic (a compound that mimics somatostatin’s actions).

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

This synonym list includes the hyphenated form SMS-201-995 for octreotide.

Research context only—not evidence of a treatment effect.

  • OCTREOTIDE
    Octreotida; Octreotide; SMS 201-995; SMS-201-995; SMS-995; SMS995
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Octreotide Long-Acting Release (OCT-LAR) is categorized as a long-acting somatostatin analog (SSA).

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

In ChEMBL, octreotide is indexed under the identifier CHEMBL1680.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Proteomics/western blotting characterization identified abundant transport-associated proteins (PIGR, MFGE8, ANXA2, CD9, CD63, CD81) in donkey-milk exosomes.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The abstract characterizes Mycapssa® as relying on transient intestinal tight-junction disruption to enhance permeability.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Physiologically, δ-cell–derived somatostatin acts as an inhibitor of pancreatic islet hormone secretion.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Octreotide is described as having pharmacological effects that may affect hemostasis, which could lower bleeding risk.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

The abstract explicitly describes the octreotide-based PET approach as SSTR-targeted PET imaging (i.e., targeting somatostatin receptors).

Research context only—not evidence of a treatment effect.

  • pubmed-42333429
    This case emphasizes an important diagnostic trap, as benign fibromatosis can mimic NET metastasis on both anatomic and SSTR-targeted PET imaging, alerting clinicians to avoid misdiagnosis and unnecessary treatment.
Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Octreotide exerts endocrine and hemodynamic actions, including suppression of growth hormone secretion and reduction of splanchnic blood flow.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Scanning electron microscopy (SEM) observations reported in the abstract indicate needle-like stearic acid features present on the mesoporous silica surface.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Characterization of exosomes isolated from donkey milk powder yielded a mean particle size of 138.4 ± 4.37 nm and a zeta potential of -42.07 ± 0.99 mV.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Radiochemical purity (RCP) for [18F]AlF-NOTA-Octreotide was reported as >95%, with stability maintained for 8 hours at room temperature, indicating the labeled octreotide tracer remained chemically intact over that period.

Research context only—not evidence of a treatment effect.

Research context · scope unclassified

1 cited source · Study independence not established

How to read this evidence

Sources and study IDs describe provenance, not clinical strength. Several articles can report the same study; one study can support several distinct findings. No clinical strength rating has been assigned here.

1 cited passage across 1 source record. 1 publication group(s) lack a resolved study identity.

Following subcutaneous administration, octreotide shows complete and rapid absorption.

Research context only—not evidence of a treatment effect.

Safety + tolerability

Risks, organized for scanning.

A structured orientation to the label—not a complete prescribing-information substitute or an individual risk estimate.

Contraindications

  • Serious hypersensitivity; additional restrictions are product-specific

Common effects

  • Gallbladder abnormalities
  • Diarrhea
  • Abdominal pain
  • Nausea
  • Injection-site pain
  • Headache

Serious risks

  • Cholelithiasis and complications
  • Glucose dysregulation
  • Bradycardia and conduction abnormalities
  • Thyroid function changes
  • Nutrient malabsorption

Structured from current product labeling [1]Regulatory labelSandostatin prescribing informationCurrent DailyMed immediate-release octreotide label.

Products + regulatory context

Same ingredient. Different records.

Brand names, routes, presentations, indications, and instructions are product-specific. This table is an index—not a substitution guide.
ProductFormProfile scopeRecord
SandostatinSubcutaneous or intravenous injectionSelected acromegaly and severe secretory diarrhea syndromes.[1]Regulatory labelSandostatin prescribing informationCurrent DailyMed immediate-release octreotide label.
Sandostatin LAR DepotLong-acting intramuscular depotMaintenance treatment in product-specific indications.[22]Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988dailymed · T1
MycapssaDelayed-release oral capsuleMaintenance treatment in selected acromegaly patients.[13]Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988dailymed · T1

Do not infer dosing, interchangeability, or an approved use from the ingredient name alone. Open the current label for the exact product and presentation.

Administration, interactions + monitoring

The practical clinical context.

Administration boundary
Subcutaneous, intravenous, intramuscular depot, or oral delayed-release depending on product. [1]Regulatory labelSandostatin prescribing informationCurrent DailyMed immediate-release octreotide label.

Research status + gaps

What still needs better answers.

A useful knowledge base names uncertainty as clearly as it names findings.
  • 1540 compiled claim(s) withheld by automated assurance: assurance_score_below_0.58 (826), assurance_score_below_0.72 (590), current_regulatory_source_required (418), evidence_scope (342), extraction_ambiguity (915), extraction_confidence_not_high (2), high_risk_requires_regulatory_or_two_independent_sources (680), no_direct_support (1408), proposal_not_staged (30)

How Peplexicon reads evidence

Authority
What kind of source is making the statement?
Independence
Do multiple citations represent separate studies—or the same evidence repeated?
Directness
Does the population, product, dose, outcome, and time horizon match the claim?
Consistency
Do credible sources support, qualify, or contradict one another?

References + discovery

Open the records yourself.

Authoritative records and published evidence are listed separately from live searches, which are discovery tools rather than pre-screened support.
  1. 1
    Regulatory labelSandostatin prescribing information

    Current DailyMed immediate-release octreotide label.

    Open ↗
  2. 2
    Literature indexEvery PubMed result for octreotide

    Live National Library of Medicine literature search; results are not pre-screened or deduplicated.

    Open ↗
  3. 3
    Trial registryEvery registered study for octreotide

    Live ClinicalTrials.gov search, including completed, active, and historical records.

    Open ↗
  4. 4
    Chemical recordoctreotide chemical record

    PubChem compound search from the National Library of Medicine.

    Open ↗
  5. 5
    Published evidence snapshotChEMBL activities for CHEMBL1680

    chembl-activities · T6

    Published 2026-08-21 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  6. 6
    Published evidence snapshotOCTREOTIDE

    chembl-molecule · T6

    Published 2026-08-21 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  7. 7
    Published evidence snapshotHIGHLIGHTS OF PRESCRIBING INFORMATIONThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-01-16 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  8. 8
    Published evidence snapshotThese highlights do not include all the information needed to use BYNFEZIA PEN safely and effectively. See full prescribing information for BYNFEZIA PEN.BYNFEZIA PEN®(octreotide acetate) injection, for subcutaneous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-02-21 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  9. 9
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-07-25 · retrieved 2026-08-28T12:18:09Z
    Open ↗
  10. 10
    Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE INJECTIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-07-15 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  11. 11
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2026-01-30 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  12. 12
    Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN INJECTION safely and effectively. See full prescribing information for SANDOSTATIN INJECTION.SANDOSTATIN®(octreotide acetate) INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2026-07-22 · retrieved 2026-08-18T22:04:15Z
    Open ↗
  13. 13
    Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-07-24 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  14. 14
    Published evidence snapshotOctreotide Acetate Injection

    dailymed · T1

    Published 2012-10-10 · retrieved 2026-08-18T22:04:11Z
    Open ↗
  15. 15
    Published evidence snapshotThese highlights do not include all the information needed to use MYCAPSSA®safely and effectively. See full prescribing information for MYCAPSSA.MYCAPSSA (octreotide) delayed-release capsules, for oral useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-07-24 · retrieved 2026-08-18T22:04:04Z
    Open ↗
  16. 16
    Published evidence snapshotRx OnlyPrescribing Information

    dailymed · T1

    Published 2018-09-21 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  17. 17
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-07-01 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  18. 18
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-07-29 · retrieved 2026-08-28T12:18:09Z
    Open ↗
  19. 19
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE injection, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-03-01 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  20. 20
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-06-25 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  21. 21
    Published evidence snapshotRx ONLY

    dailymed · T1

    Published 2019-01-07 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  22. 22
    Published evidence snapshotThese highlights do not include all the information needed to use SANDOSTATIN LAR DEPOT safely and effectively. See full prescribing information for SANDOSTATIN LAR DEPOT.SANDOSTATIN®LAR DEPOT (octreotide acetate) for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2025-12-22 · retrieved 2026-08-18T22:04:06Z
    Open ↗
  23. 23
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-05-23 · retrieved 2026-08-28T12:18:09Z
    Open ↗
  24. 24
    Published evidence snapshotThese highlights do not include all the information needed to useOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSIONsafely and effectively. See full prescribing information forOCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATEfor injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-07-30 · retrieved 2026-08-18T22:04:08Z
    Open ↗
  25. 25
    Published evidence snapshotOctreotide Acetate Injection

    dailymed · T1

    Published 2012-10-10 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  26. 26
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE FOR INJECTABLE SUSPENSION.OCTREOTIDE ACETATE for injectable suspension, for gluteal intramuscular useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2026-01-21 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  27. 27
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-05-07 · retrieved 2026-08-25T11:03:05Z
    Open ↗
  28. 28
    Published evidence snapshotThese highlights do not include all the information needed to use OCTREOTIDE ACETATE INJECTION safely and effectively. See full prescribing information for OCTREOTIDE ACETATE INJECTION.OCTREOTIDE ACETATE INJECTION, for subcutaneous or intravenous useInitial U.S. Approval: 1988

    dailymed · T1

    Published 2024-12-03 · retrieved 2026-08-28T12:18:09Z
    Open ↗
  29. 29
    Published evidence snapshotOctreotide Acetate Long-Acting Formulation Versus Open-Label Subcutaneous Octreotide Acetate in Malignant Carcinoid Syndrome

    doi · T6

    Published 1999-02-01 · retrieved 2026-09-09T18:01:34Z
    Open ↗
  30. 30
    Published evidence snapshotIUPHAR ligand commentary

    iuphar-comments · T6

    Published 2026-08-24 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  31. 31
    Published evidence snapshotIUPHAR interactions for octreotide

    iuphar-interactions · T6

    Published 2026-08-24 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  32. 32
    Published evidence snapshot[<sup>67</sup>Ga]NODAGA-[Tyr<sup>3</sup>]octreotide

    iuphar-ligand · T6

    Published 2026-08-21 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  33. 33
    Published evidence snapshotOctreotide acetate long-acting formulation versus open-label subcutaneous octreotide acetate in malignant carcinoid syndrome.

    pubmed · T2

    Published 1999-02-01 · retrieved 2026-09-09T18:01:33Z
    Open ↗
  34. 34
    Published evidence snapshotMega-dose intravenous octreotide for the treatment of carcinoid crisis: a systematic review.

    pubmed · T2

    Published 2013-05-01 · retrieved 2026-09-09T22:30:04Z
    Open ↗
  35. 35
    Published evidence snapshotDebut of a somatostatin analog: octreotide in review.

    pubmed · T3

    Published 1989-12-01 · retrieved 2026-09-09T22:30:03Z
    Open ↗
  36. 36
    Published evidence snapshotOctreotide. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in conditions associated with excessive peptide secretion.

    pubmed · T3

    Published 1989-11-01 · retrieved 2026-09-08T10:56:07Z
    Open ↗
  37. 37
    Published evidence snapshotOral Octreotide: A Review of Recent Clinical Trials and Practical Recommendations for Its Use in the Treatment of Patients With Acromegaly.

    pubmed · T3

    Published 2022-06-01 · retrieved 2026-09-09T22:30:04Z
    Open ↗
  38. 38
    Published evidence snapshotOctreotide Subcutaneous Depot for Acromegaly: A Randomized, Double-blind, Placebo-controlled Phase 3 Trial, ACROINNOVA 1.

    pubmed · T2

    Published 2025-05-19 · retrieved 2026-09-08T21:45:41Z
    Open ↗
  39. 39
    Published evidence snapshotComprehensive design and characterization of pH-gradient-loaded donkey-milk exosomes for oral octreotide delivery: A bench-to-in silico roadmap.

    pubmed · T3

    Published 2026-04-25 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  40. 40
    Published evidence snapshotFunctionalised mesoporous silica with stearic acid: A novel approach to improve octreotide delivery.

    pubmed · T3

    Published 2026-04-25 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  41. 41
    Published evidence snapshotAnti-secretory and anti-proliferative actions of next-generation dual subtype 2 and 5 somatostatin receptor ligands in neuroendocrine tumor models.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-05T09:00:33Z
    Open ↗
  42. 42
    Published evidence snapshotDual-tracer PET/CT and cocktail therapy with [177Lu]Lu-FAP2286 and [177Lu]Lu-DOTATATE in G3 Neuroendocrine Tumors (NET).

    pubmed · T3

    Published 2026-07-01 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  43. 43
    Published evidence snapshotReal-World Observational Study of Somatostatin Analogs and Rescue Medication Usage for Neuroendocrine Tumors in Canada.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-04T22:24:53Z
    Open ↗
  44. 44
    Published evidence snapshotSSTR2-targeting therapy in EBV-positive and EBV-negative metastatic nasopharyngeal carcinoma.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  45. 45
    Published evidence snapshotCongenital Hyperinsulinism in Neonates: Diagnostic Challenges and Management in Two Cases With KCNJ11 and ABCC8 Mutation.

    pubmed · T3

    Published 2026-02-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  46. 46
    Published evidence snapshot[Optimal timing for octreotide administration in adult patients with chylothorax: A scoping review].

    pubmed · T3

    Published 2026-06-16 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  47. 47
    Published evidence snapshotPulmonary neuroendocrine tumour-associated ectopic Cushing's syndrome: diagnostic challenges and multidisciplinary management.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  48. 48
    Published evidence snapshotEffect of octreotide-deoxycholate hydrophobic ion pairing solid dispersions on intestinal permeability to enhance octreotide absorption via increased lipophilicity and ASBT-mediated transport.

    pubmed · T3

    Published 2026-05-05 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  49. 49
    Published evidence snapshotMedical Versus Surgical/Endoscopic Management of Malignant Bowel Obstruction in Patients With End-Stage Gynecologic Cancer: A 12-Year Single-Center Experience.

    pubmed · T3

    Published 2026-02-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  50. 50
    Published evidence snapshotMidodrine Monotherapy in Refractory Hepatorenal Syndrome-Acute Kidney Injury: A Case Report.

    pubmed · T3

    Published 2026-02-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  51. 51
    Published evidence snapshotThe management of hepatorenal syndrome-acute kidney injury (HRS-AKI): A national survey of hepatology provider practices.

    pubmed · T3

    Published 2026-04-01 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  52. 52
    Published evidence snapshotPrimary Intestinal Lymphangiectasia Presenting as Recurrent Chylous Ascites: A Rare Case.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  53. 53
    Published evidence snapshotSSTR2 expression in EBV-positive and EBV-negative lymphomas.

    pubmed · T3

    Published 2026-04-10 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  54. 54
    Published evidence snapshotWhat is the future of acromegaly therapy?

    pubmed · T3

    Published 2026-06-04 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  55. 55
    Published evidence snapshotDevelopments in Pharmacotherapy for Acromegaly: Current and Emerging Approaches.

    pubmed · T3

    Published 2026-06-01 · retrieved 2026-08-28T12:18:09Z
    Open ↗
  56. 56
    Published evidence snapshotOctreotide for prevention of delayed bleeding after endoscopic mucosal resection for large superficial non-ampullary duodenal tumors.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  57. 57
    Published evidence snapshotA 13-Year-Old Girl with Congenital Hyperinsulinemic Hypoglycemia Due to anABCC8Mutation and Recent Onset of Diabetes Mellitus: A Case Report and Literature Review.

    pubmed · T3

    Published 2026-04-14 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  58. 58
    Published evidence snapshotIdentification and Localization of Functioning Gastroenteropancreatic Neuroendocrine Tumors Using [18F]F-NOTA-octreotide PET/CT.

    pubmed · T3

    Published 2026-03-31 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  59. 59
    Published evidence snapshotOptimization of automated radiosynthesis method for [18F]AlF-NOTA-Octreotide and PET/CT imaging in neuroendocrine neoplasms.

    pubmed · T3

    Published 2026-04-21 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  60. 60
    Published evidence snapshotUptake of18F-AlF-NOTA-octreotide PET/CT in gastrointestinal stromal tumors.

    pubmed · T3

    Published 2026-04-24 · retrieved 2026-09-01T08:37:10Z
    Open ↗
  61. 61
    Published evidence snapshotpubmed-42029102

    pubmed · T3

    Published 2026-08-17 · retrieved 2026-08-17T23:10:15Z
    Open ↗
  62. 62
    Published evidence snapshotUpdate on PET Imaging of Neuroendocrine Neoplasms.

    pubmed · T3

    Published 2026-06-01 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  63. 63
    Published evidence snapshotComparison of [111In]octreotide Scintigraphy and [68Ga]DOTATOC PET in Gastroenteropancreatic Neuroendocrine Tumors: Concordance of Krenning Scores and Implications for Peptide Receptor Radionuclide Therapy Eligibility.

    pubmed · T3

    Published 2026-06-12 · retrieved 2026-08-24T17:38:00Z
    Open ↗
  64. 64
    Published evidence snapshotAmino acids partially override inhibitory effects of octreotide on islet hormone secretion in healthy individuals.

    pubmed · T3

    Published 2026-07-01 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  65. 65
    Published evidence snapshotEvaluation of [¹⁸F]AlF-NOTA-octreotide PET/CT in routine clinical use: a retrospective analysis in 288 neuroendocrine tumor patients.

    pubmed · T3

    Published 2026-09-01 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  66. 66
    Published evidence snapshotpubmed-42333429

    pubmed · T3

    Published 2026-08-17 · retrieved 2026-08-17T23:10:15Z
    Open ↗
  67. 67
    Published evidence snapshotSpinal phosphaturic mesenchymal tumor: a case report of thoracic vertebral involvement with preoperative embolization and literature review.

    pubmed · T3

    Published 2026-07-03 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  68. 68
    Published evidence snapshotpubmed-42442014

    pubmed · T3

    Published 2026-08-17 · retrieved 2026-08-17T23:10:15Z
    Open ↗
  69. 69
    Published evidence snapshotComparative Efficacy and Safety of Octreotide, Lanreotide, and Pasireotide in ADPKD and PLD: A Network Meta-analysis with Real-world Evidence from the FAERS Database.

    pubmed · T3

    Published 2026-07-20 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  70. 70
    Published evidence snapshotEx Vivo drug sensitivity in patient-derived 3D cultures in acromegaly and its association with clinical predictors.

    pubmed · T3

    Published 2026-07-24 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  71. 71
    Published evidence snapshotImpact of dosage form on the pharmacokinetics of octreotide after oral administration with permeation enhancers.

    pubmed · T3

    Published 2026-09-05 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  72. 72
    Published evidence snapshotEfficacy and Safety of Octreotide for Gastrointestinal Bleeding Due to Portal Hypertension in Children-A Systematic Review.

    pubmed · T3

    Published 2026-06-24 · retrieved 2026-08-24T17:18:21Z
    Open ↗
  73. 73
    Published evidence snapshotAnalysis of outcome in patients with different primary localisation of neuroendocrine tumors after PRRT. 10 years single institution experience.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  74. 74
    Published evidence snapshotGhrelin and relamorelin counteract hypoglycemia in mice engrafted with congenital hyperinsulinism stem cell-derived islets.

    pubmed · T3

    Published 2026-07-20 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  75. 75
    Published evidence snapshotSolitary left frontotemporal neuroendocrine metastasis mimicking a high-grade astrocytoma.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-08-21T17:03:42Z
    Open ↗
  76. 76
    Published evidence snapshotMultiple skin and subcutaneous metastasis as initial manifestation in neuroendocrine carcinoma lung: A rare case report.

    pubmed · T3

    Published 2026-10-01 · retrieved 2026-08-17T23:10:15Z
    Open ↗
  77. 77
    Published evidence snapshotStructural control and resilience in the oxytocin molecular graph: A graph-theoretic framework for critical atom and bond identification with comparative validation across cyclic peptides.

    pubmed · T3

    Published 2026-11-01 · retrieved 2026-09-07T08:44:20Z
    Open ↗
  78. 78
    Published evidence snapshotEditorial: Toward Prognostic Precision in the Management of Gastroenteropancreatic Neuroendocrine Neoplasms.

    pubmed · T3

    Published 2026-01-01 · retrieved 2026-09-09T08:36:24Z
    Open ↗
  79. 79
    Published evidence snapshotpubmed-42604001

    pubmed · T3

    Published 2026-08-17 · retrieved 2026-08-17T23:10:15Z
    Open ↗
  80. 80
    Published evidence snapshotThe role of biorelevant media components on the diffusion and enzymatic stability of oral cyclic peptide analogs.

    pubmed · T3

    Published 2026-09-04 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  81. 81
    Published evidence snapshotAssessment of Neuroendocrine Features Using 99mTc-Octreotide Scintigraphy in Patients with Metastatic Castration-Resistant Prostate Cancer: Does it Predict Response to 177Lu-PSMA Radioligand Therapy?

    pubmed · T3

    Published 2026-08-29 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  82. 82
    Published evidence snapshotOctreotide Administration Methods in Sulfonylurea Poisoning: A Retrospective Chart Review.

    pubmed · T3

    Published 2026-09-02 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  83. 83
    Published evidence snapshotDifferential Somatostatin Sensitivity of Corticotropic and Somatotropic Responses Following Amino Acid Infusion.

    pubmed · T3

    Published 2026-09-04 · retrieved 2026-09-05T08:43:42Z
    Open ↗
  84. 84
    Published evidence snapshotClinical effects of octreotide compared to placebo in patients with gastrointestinal neuroendocrine tumours. Report on a double-blind, randomized trial.

    pubmed · T2

    Published 1995-03-01 · retrieved 2026-09-08T21:46:11Z
    Open ↗
  85. 85
    Published evidence snapshotSomatostatin and somatostatin analogues: pharmacokinetics and pharmacodynamic effects.

    pubmed · T3

    Published 1994-01-01 · retrieved 2026-09-09T18:03:34Z
    Open ↗
  86. 86
    Published evidence snapshotSandostatin LAR (microencapsulated octreotide acetate) in acromegaly: pharmacokinetic and pharmacodynamic relationships.

    pubmed · T3

    Published 1996-08-01 · retrieved 2026-09-08T21:46:09Z
    Open ↗